Mianserin

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CAS: 24219-97-4

Name:

Mianserin

Other names:

Mianserine; Mianserina; Mianserinum; Tolvon; Mianseryna [Polish]; Mianseryna; Norval; Mianserine [INN-French]

A tetracyclic compound with antidepressant effects. Mianserin was previously available internationally, however in most markets it has been phased out in favor of Mirtazapine.

Interactions

Description

UniProt ID

Protein: Muscarinic acetylcholine receptor, Gene: CHRM1
Protein: Muscarinic acetylcholine receptor, Gene: CHRM2
Protein: Muscarinic acetylcholine receptor M3, Gene: CHRM3
Protein: Muscarinic acetylcholine receptor M4, Gene: CHRM4
Protein: Muscarinic acetylcholine receptor M5, Gene: CHRM5
Protein: Alpha-1A adrenergic receptor, Gene: ADRA1A
Protein: Alpha-1B adrenergic receptor, Gene: ADRA1B
Protein: Alpha-1D adrenergic receptor, Gene: ADRA1D
Protein: Alpha-2A adrenergic receptor, Gene: ADRA2A
Protein: Alpha-2B adrenergic receptor, Gene: ADRA2B
Gene: ADRA2C
Protein: D(1A) dopamine receptor, Gene: DRD1
Protein: D(2) dopamine receptor, Gene: DRD2
Gene: DRD3
Protein: D(4) dopamine receptor, Gene: DRD4
Protein: Sodium-dependent dopamine transporter, Gene: SLC6A3
Protein: Sodium- and chloride-dependent GABA transporter 2, Gene: SLC6A13
Protein: ATP-dependent RNA helicase DHX8, Gene: DHX8
Protein: Histamine H2 receptor, Gene: HRH2
Protein: Histamine H3 receptor, Gene: HRH3

Toxicity

oral LD50 [mouse] mg/kg
Unavailable
oral LD50 [rat] mg/kg
> 780.0
oral LD50 [rabbit] mg/kg
Unavailable

Effects on organism

Anti Inflammation
Anti Depressant
Antibacterial

No

Antifungal

No

Antiviral

No

Longevity mechanisms activation

Calorie Restriction Mimetics
+
Stress Resistance
+

Suppression of aging mechanisms

No data

Relation to biomarkers of Aging

Data not available

Relation to aging associated genes

No data available

Experimental conditions

liquid medium + E. coli OP50

Life Extension

Mean LS (%)
32.0
Median LS (%)
Mortality rate derease (%)
Max LS (%)
Cell CLS
Cell RLS

Concentration wth maximum effect

50 mkM

More info about experiment

18033297 24134630
Opposite effect19112515