Guanabenz Acetate

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CAS: 23256-50-0

Name:

Guanabenz Acetate

Other names:

Wytensin; Guanabenz acetate; Guanabenz monoacetate; Acetate; Guanabenz; Monoacetate; Wy 8678; Wy-8678

Guanabenz acetate is an α2A-AR adrenergic agonist and IGRS (imidazoline I2 binding site) selective ligand. Guanabenz acetate is an activator of alpha2B-AR (α2b-adrenergic receptor) and alpha2C-AR (α2c-adrenergic receptor).

Interactions

Description

UniProt ID

Protein: Alpha-2A adrenergic receptor, Gene: ADRA2A
Protein: Alpha-2B adrenergic receptor, Gene: ADRA2B
Protein: 5-hydroxytryptamine receptor 1A, Gene: HTR1A
Protein: Amine oxidase [flavin-containing] A, Gene: MAOA
Protein: Amine oxidase [flavin-containing] B, Gene: MAOB
Protein: Nanos homolog 1, Gene: NANOS1

Toxicity

oral LD50 [mouse] mg/kg
Unavailable
oral LD50 [rat] mg/kg
> 238.0
oral LD50 [rabbit] mg/kg
Unavailable

Effects on organism

Anti Inflammation
Neuroprotective
Cardioprotective
Antibacterial

No

Antifungal

No

Antiviral

No

Longevity mechanisms activation

Stress Resistance

Suppression of aging mechanisms

Anti Oxidant
+

Relation to biomarkers of Aging

Antihypertensive therapy

1686570 6148885

Relation to aging associated genes

No data available

Experimental conditions

S-complete media in wells of 96 well + E. coli OP50plates containing E. coli OP50

Life Extension

Mean LS (%)
12.0
Median LS (%)
Mortality rate derease (%)
Max LS (%)
Cell CLS
Cell RLS

Concentration wth maximum effect

0,33%

More info about experiment

24134630
Opposite effectNo