Buformin

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CAS: 692-13-7

Name:

Buformin

Other names:

1-Butylbiguanide; Buformine; Butylbiguanide; Butylbiguanidum; Butyldiguanide; Butformin; Glybigid; Glybigidum; Adebit

Buformin is an anti-diabetic drug of the biguanide class, chemically related to metformin and phenformin. It was withdrawn from the market in most countries due to a high risk of causing lactic acidosis.

Interactions

Description

UniProt ID

Protein: Glutathione-specific gamma-glutamylcyclotransferase 1, Gene: CHAC1
Protein: Solute carrier family 22 member 2, Gene: SLC22A2
Protein: Tumor necrosis factor receptor superfamily member 1A, Gene: TNFRSF1A

Toxicity

oral LD50 [mouse] mg/kg
Unavailable
oral LD50 [rat] mg/kg
Unavailable
oral LD50 [rabbit] mg/kg
Unavailable

Effects on organism

Anti Cancer
Anti Diabetic
Antibacterial

No

Antifungal

No

Antiviral

No

Longevity mechanisms activation

No data

Suppression of aging mechanisms

No data

Relation to biomarkers of Aging

Improved insulin sensitivity

15533580

Relation to aging associated genes

No data available

Experimental conditions

Not available

Life Extension

Mean LS (%)
Median LS (%)
23.5
Mortality rate derease (%)
Max LS (%)
26.1
Cell CLS
Cell RLS

Concentration wth maximum effect

More info about experiment

Bakaev VV (2002. Effect of 1-butylbiguanide hydrochloride on the longevity in the nematoda Caenorhabditis elegans. Biogerontology 3 (Suppl 1): 23–24
Opposite effectNo

Experimental conditions

Not available

Life Extension

Mean LS (%)
7.3
Median LS (%)
Mortality rate derease (%)
Max LS (%)
5.5
Cell CLS
Cell RLS

Concentration wth maximum effect

5 mg/rat/day

More info about experiment

14618027
Opposite effectNo