2-Deoxy-D-Glucose

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CAS: 154-17-6

Name:

2-Deoxy-D-Glucose

Other names:

2-Deoxy-D-arabino-hexose; SMR000857164; Ba 2758, 2-dGlc; SureCN7669; D-Arabino-2-deoxyhexose; Deoxyglucose

2-Deoxy-D-glucose is an apoptosis inhibitor that has been shown to be taken up by glial cells incubated with insulin. Studies indicate that this compound has the potential to suppress hypoxia in murine retinal tissue. Additionally, 2-Deoxy-D-glucose has been noted to be a glycolytic inhibitor via indirect inhibition of hexokinase (HXK) which results in endoplasmic reticulum stress. Other experiments suggest that this agent upregulates autophagy and lowers ATP levels in certain cancer cell lines. 2-Deoxy-D-glucose is an activator of AMPK and an inhibitor of GPI.

Interactions

Description

UniProt ID

Protein: 5'-AMP-activated protein kinase catalytic subunit alpha-1, Gene: PRKAA1
Protein: 5'-AMP-activated protein kinase catalytic subunit alpha-2, Gene: PRKAA2

Toxicity

oral LD50 [mouse] mg/kg
Unavailable
oral LD50 [rat] mg/kg
Unavailable
oral LD50 [rabbit] mg/kg
Unavailable

Effects on organism

Anti Convulsant
Neuroprotective
Antibacterial

No

Antifungal

No

Antiviral

No

Longevity mechanisms activation

Hormetin
Calorie Restriction Mimetics
Stress Resistance

Suppression of aging mechanisms

No data

Relation to biomarkers of Aging

Increased intracellular NAD(+) levels in both time- and concentration-dependent manners. 2-DG also dose-dependently increased SIRT1 activities and the lifespan (measured as the cumulated growth curve of population doubling levels) of Hs68 cells; Suppress the level of constitutive mTOR- and DNA damage- signaling.

21604001 23363784 24677687

Relation to aging associated genes

No data available

Experimental conditions

Not available

Life Extension

Mean LS (%)
17.0
Median LS (%)
Mortality rate derease (%)
Max LS (%)
25.0
Cell CLS
Cell RLS

Concentration wth maximum effect

5 mM

More info about experiment

17908557
Opposite effectNo

Experimental conditions

Not available

Life Extension

Mean LS (%)
Median LS (%)
Mortality rate derease (%)
Max LS (%)
-10.0
Cell CLS
Cell RLS

Concentration wth maximum effect

0.25%

More info about experiment

Opposite effect20026095